Hauora, Mau faaineineraa
"Propranolol": analogues, tohutohu mo te whakamahi, whakaahuatanga me arotake
"Propranolol" - he rongoā no ki te rōpū o blockers whiriwhiri. He pānga antianginal, antiarrhythmic me hypotensive te tarukino. Ko te medicament whakahaeretia mo te whakaaro o te maimoatanga o te manawa toto pūroto, thyrotoxicosis, takawhita. he whai hua i roto i te rongoā neuro dystonia, migraine. Kei te whakamahia te reira i roto i te whakatinanatanga o te maimoatanga o te kore ngakau, pectoris angina. whai hua te tarukino te tinana i roto i te infarction myocardial. hamani ratou arrhythmia me cardiomyopathy hypertrophic. A, no te kahore he tika te manawanui e whakaaro "Propranolol" ritenga he kaitūtohu mātanga e mo te manawanui ko te tino pai.
Puka tuku
Ka taea e koe te hoko e rua ngā momo o te tarukino - tarukino "Propranolol" me te tarukino "Propranolol Nycomed". Ko te taua rongoa e kua whakaputaina e kamupene rerekē i roto i te papa tenei.
Ko te wāhanga o te tarukino
hanga te faaineineraa i runga i te pūtake o te taonga propranolol kaha. Horopeta kia rerekē wāhanga matua - 10, 40, 80 me te 160 mg i roto i te hanganga o ia papa.
He rerekē kai Ngaahi Houalotú whakamahia i roto i te hanga o papa, me whakawhirinaki i runga i nga kaihanga. Hei mohio rite te mea kei roto i te rongoā i mua i te whakamahi i te mea e tika ana ki te pānui i te buka haapiiraa.
Ko te pānga haumanu o te tarukino
He whakaatu i te kaha ki te ārai i te mau farii ohipa beta-adrenergic tikanga "Propranolol" ako ā-ringa. Analogues i runga i te tinana rite ki te mahi. pā Papa i iaia receptors peta taiepa 1 me 2. Ko te pānga inhibitory i runga i enei receptors arata'i ki te whakangā o taiepa iaia, ai whakakore tokomaha o nga raruraru - pēhanga toto tiketike, nui haere te hiahia cardiac mō te whiwhi hāora, supply rawakore o ngā matūkai me te hāora ki te kopa, i nga okana.
mahi Antiarrhythmic o te raau taero whakatairanga te ahua o ngā rerekētanga pai i roto i te tinana, pērā i te automaticity māori pakohu kōpuku, whakaiti āriponga kōpuku atrioventricular, whakakorenga o nui haere excitability o ngā pūtau e Kei roto i te myocardium. Ngā mihi ki te "Propranolol" whakahokia mahi noa o te ngakau, i reira he kahore tauhohenga ki akiaki waho, pēhia kia e pā tona manawataki.
whakatairanga "Propranolol" analogues te whanaketanga o te pānga anti-anginal e whakaaturia ake āhua o uaua cardiac, te whakaiti i te nui o te hāora e hiahiatia mo tona mahi. Tenei te tikanga e titau te ngakau iti hāora ki te kia heke, ka heke i te auautanga o enei contractions te rawa.
hāngai ana mahi Hypotensive te i runga i te hua i roto i te lumen o oko toto, me te whakangā o ratou taiepa. Taupānga o te horopeta kotahi o papa arata'i ki te whakaiti o te pēhanga toto, puritia te pānga hua te hoki i te iti rawa 20 haora te pō. kitea pānga hypotensive pūmau i muri i rua wiki o te whakamahi auau o pire. e kore te mea e tika ana mo te tanga o ngā āhuatanga tahi e te hua koi i roto i te pēhanga te tarukino, kua tohua i te reira no te therapy wā roa-no te takawhita.
whakamahi wā-roa taero arata'i ki te whanaketanga o ngā pānga cardioprotective. Whakaaturia te hekenga i roto i te tūponotanga o te hohokitanga o infarction myocardial i muri i te tikanga o taua therapy "Propranolol" arotake, tohutohu. Tino heke te mōrea o te mate ohorere puta. Kei te mohiotia te reira e te raau he pānga pai i te pēhanga intraocular faateiteihia.
Pharmacokinetics
I muri whiwhi roto te wahi matua tinana whenumi te tarukino (e pā ana ki 90%), i te mea kei hokiate te taupū o te bioavailability. Communication ki pūmua ōrite ana ki 93%. nekehia Drug i te tinana kei i te mimi, e hinga metabolites. momo tamau kua iti iho i te kotahi ōrau o te rongoā.
iteraa papû
taea "Propranolol" ako analogues ki a koutou tautapa i te maimoatanga o etahi tikanga me mate. Ratou tukinotia takawhita portal, me te matua, te ma'ii'o myocardial, hyperthyroidism. tauturu rongoā noho te huru i te lumen whāiti o te haoraora, faaati faufaa, patua aitua, e taea te whakamahi rite te taputapu mo te whakamahi i roto i te prophylaxis o migraine. Papa e tika ana mō te therapy i roto i te ngakau o te hoia, infarction myocardial, arrythmia. Kei te whakahaere te tarukino ki tūroro ki prolapse takirere mitral. Na roto i te tohu ngā tachycardia supraventricular me te pakohu. Vahe tikanga whakamana i te syndrome withdrawal, pectoris angina, akathisia, puta tika ki te whakamahi o neuroleptics. Rongoā whakaritea ki tūroro ki pheochromocytoma mō huinga therapy. whakamahia te raau i roto i te ngoikore o te mahi mahi i muri i menopause ki te whakakore ona faaiteraa kino.
contraindications
Vai nei te tahi contraindications mō "Propranolol" tarukino. Ka taea te tīpakohia Analogs i roto i te wā i reira e kore e he e tika ana te tarukino. Contraindications ngā:
- tikanga ātete wāhanga;
- ru cardiogenic;
- bradycardia, i roto i nei te maha o heartbeats ia meneti ko 55 sp.;
- acidosis pūkoro;
- kore ngakau ma'i ranei puka whakapeka;
- vasomotor Rhinitis;
- poraka sinoatrial, atrioventricular (2, tohu 3);
- Prinzmetal angina ;
- pēhanga toto iti;
- Whakamahia o taiāki huka;
- syndrome tahi e te pakohu;
- wā aroaro i roto i nei te nohopuku auroa reira;
- raruraru ki te tohanga piringa (decompensation taahiraa);
- mate arata'iraa whakawhiti i mua i roto i nei pānga Airways, huangō, bronchospasm wātea.
He hoki ngā āhuatanga i reira e hiahiatia tūpato te. I roto i te wā e whai ake nei, ka taea e koe te whiriwhiri hei utu o te tarukino "Propranolol" analogues, taurite:
- gravis myasthenia;
- mate huka (decompensated, subcompensation);
- uaua cardiac iti hoki (huangō), ate, whatukuhu;
- colitis mate hukihuki;
- korekore;
- poraka atrioventricular (tohu tuatahi);
- psoriasis;
- nui haere mahi o te repe thyroid;
- momo ma'i o Bronchitis;
- huka toto iti;
- emphysema;
- koroheketanga;
- I roto i te hapū, breastfeeds.
maimoatanga tarukino
Tūroro ki te takawhita kia tangohia horopeta tarukino rua rā o 40 mg ia horopeta kotahi. Ko taea tona hua i roto i 14-28 ra. Ki te tika, ka taea e papa te inu ia i roto i te inenga o te 80 ki te 160 mg. Ko te auau o te tikanga te whiwhi ko te taua.
A, no te inu e toru ranei e wha nga wa ia tachyarrhythmia tūroro pakeke i te 10 ki te 30 mg ia fariiraa "propranolol" tikanga. Ka taea te whakamahi Analogs, ki te kore tenei hua e uru. tūroro e Si◊í ki te raruraru taua o te tarukino faaterehia i roto i te nui o i 0.2 ki te 0.4 mg ia taimaha tinana kirokaramu. Ko te auau o te tono tikanga - rite toru ranei wha nga wa he ra.
Ka rite ki te mehua ārai i roto i tūroro e kua tāutuhia angina whakarite wha tango i tenei rongoā katoa ra. He horopeta kotahi o te 20 mg. Ko taea tona hua mō te whitu nga ra. tangohia 40 mg o tarukino te i te auau taua, 80 mg - paku iti maha (rua).
I muri prophylaxis infarction myocardial hiahiatia. Rere taea medicament reira "Propranolol". Rahi tika horopeta kotahi ko 40 mg, kia te pōhiri tarukino ia ra kia whakahaerea e toru. Whakanuia te horopeta noa te mōrahi o 80 mg.
Me tutaki āraihia migraine ki te whakamahi o 40 mg o te tarukino rua he ra. Hiahia he hua i roto i te horopeta ki 80 mg, tango rongoā ia kia kia tokorua ranei e toru, me nga tamariki - e toru ranei wha. Tātaitanga o te horopeta mō ngā tūroro ki te iti whakamana i roto i te whakaaro o to ratou taimaha, ia manokaramu o - i 1.5 ki te 2 mg.
Thyrotoxicosis - he mate i roto i i homai te tarukino te 10 mg engari e kore e neke atu i te 40 mō te fariiraa i toru ranei e wha nga wa he ra.
Ki te whakamahere koe ki pheochromocytoma therapy, ngā te raau e ki te blockers alpha.
pānga taha
Me whakarongo ki te mea whakatau te pānga taha o raau taero "Propranolol" ā-ako. Analogs arotake - e kore he kōrero iti nui, awe te pai rawa o ngā rongoā mō te maimoatanga. Ki he iti te mōrea o tauhohe kino o te tinana, he mea e tika ana ki te āta pānui i te tohutohu, he reira pai ki te kia maheni ki.
Rongoā, ki te whakamahia hē e taea kino i te pūnaha Cardiovascular meinga e raruraru i roto i te pūnaha io pokapū, te pūnaha endocrine. faaiteraa kino pea i runga i te wahi o te wahi kūnatu, kia whakakorikoria nga kiriuhi mucous me kiri. I roto i te pānga taha tabulahia i roto i te tohutohu - raruraru romahā. He kia kia atu ngā pānga taha.
utu Analogs
I mua i te hoko "Propranolol" analogues tarukino, kua maha ako te utu tūroro. Hokona pire e taea kia hoki 16-75 moni. whakaritea Price e te maha o papa ia mōkihi. Whakakapia taea te tarukino e "Propranobene" medicaments "obzidan" ranei "Inderal". Ka taea hoki te hanga e koe te maimoatanga "Inderalom LA", "Inderalom".
Na roto i te tohutoro ki te tarukino "Propranolol" tohutohu mō te whakamahi, utu, whakarato analogs mōhiohio nui e tauturu hanga i te whakatau pai ka kōwhiri rongoā me maimoatanga.
Reviews
Reviews te nuinga pai. korerotia ratou e ko maha whai hua te maimoatanga tarukino. I tua atu, he tokomaha e makona ki te rongoa utu iti. "Propranolol" whakahaere ki te pupuri i te pēhanga toto i te taumata noa, hohoro te too atu o palpitations ngakau. Rongoā whakaiti tohu o te mate ngakau, faaore kare tangata. arotake tōraro e te nuinga o waiho te iwi no te mea o ngā pānga taha mamafa e kia puta i roto i therapy. I te tahi taime i reira he ngoikore nui, raruraru moe, ri'ari'ai.
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