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Tohutohu mō te whakamahi, hei tairitenga "Cefotaxime" me arotake

"Cefotaxime" (tohu mo te whakamahi, te ture mō te tātai i te inenga tino pai, me te te analogues tino rongonui ka hoatu i raro nei) ko te rongoā paturopi āhua-waihanga hou. he ātete ki te beta-lactamases reira me he kaha ki e rua karamu-pai, me te karamu-kino microorganisms. Tikanga tauhohenga matüora tika ki te pehanga o te kaha o ngā wāhanga o ngā tukanga māori puta i roto i te membrane pūtau o tukumate.

Te raau e whiwhi ki roto ki te tinana, āta e whakamotitia te peptidoglycan hononga cruciform, kia tika hoki ki nga huakita whakarite te noho pūmau o te taiepa tūturu. Ka rite ki mohiotia te, paturopi me inhibitors kai te kaipahua, rapa pūtau - he āhua ngāwari ūnga tenei.

Puka tuku

Ko te medicament "Cefotaxime" (werohanga ā-me infusions he hakari rite anake te ara iahiko tuku taea o te taonga kaha) e tukua ki te mākete ho'oraa i roto i te puehu ma kowhai ranei, e te kaimahi rite pūtake mō te faaineineraa o te otinga. Ko te ampoules werohia pera-ka karanga tenei.

Ko te taketake 10 oko rōrahi ml hanga o te karaihe piata. Te hakari papatipu kaiwhakahohe tūturu i roto i te kōwae hua taua tei runga i te whakakī o te kopu (0.5, 1.0 2.0 karamu ranei).

tauari pharmacokinetic

tonu kia tuhia te reira e kore nga tairitenga "Cefotaxime" kua te āhuatanga pharmacokinetic taua rite te taketake. I roto i ngā, ki te kōrero tatou e pā ana ki te auau o te absorption o wāhanga i te wāhi i werohia, te mimititanga o enei āpiha, te whakawa i nga kōrero o ngā maha, he reira nui tere atu i te absorption tuatahi o te taua tonu "Duataksa" ranei "Tsetaksa". "Tītohunga" takoto te take i roto i te hanganga tauira rāpoi ngota tuatahi. Tohunga i roto i ta ratou mau pahonoraa fakamamafa'i te meka e Kei roto i te kano Indian i runga "poke ho'oraa" i roto i te puka o pärönaki cephalosporin matatini e tino pōturi te pākia o te tahi atu kai.

Kei te kitea te reira e "Cefotaxime" (pānuitanga tohutohu i roto i te aratohu e pā ana ki te tarukino hoatu, faaore i te tūponotanga o te ūnga i te aroaro o te toto) whakaaturia te taumata āhua teitei o here ki pūmua wē, i rerekē te roanga o te pānga microbicidal i roto i 11-12 haora. He he kaihoko panoni tīmata te whakanoho tohaina i roto i te tinana, tae atu wheua (te kitea hoki kukū mōrahi i roto i te myocardium me te tōngāmimi kawa).

Ko te whakauru matua o te mea i kaha i te arai placental me riro te wāhi o te pericardium me inu cerebrospinal. e kore e nui ake te toharite hawhe-ora o te whaowhia te maturuturunga iho rō-uaua kotahi haora ki te werohanga intramuscular - kotahi meneti rau-waru tekau. e kore te Tetahi o whāiti te haaputuputuraa o te rauemi tohua - wahi o te wāhanga tahi excreted te i roto i te ate, me te tahi atu (e pā ana ki 90%) - mimi. I roto i te take whakamutunga, te rahi o metabolites kaha iti ki 20-30% o te horopeta faaterehia, i.e. e pā ana ki 70% o te otinga mahue te tinana, kahore pangia whakarerekētanga hanganga.

Tuhinga hoki

Kei te pai te whakapumautia enei māngai rite te pūārai o ngā tukanga hopuhopu, me te inflammatory rere microorganisms, ngā tairongo ki cefotaxime. Na taunakitanga o tenei ko kore anake rangahau haumanu - ka taea te hanga mutunga rite i muri i te tai'oraa i te maha arotake pai whakairi ki runga ki te pae tukutuku, te kaupapa o nei ko te tarukino whai hua ki te whawhai tukumate. Front mahi pharmacological o te tarukino i makona whanui, engari atu pinepine "i runga i te titiro" hinga ma'i ranei whakapeka disorders tākihi puta me te mimi, me te mate romahā o runga.

Me ahau mea e, ara, ki te te tuakiri tino o te hanganga o te tairitenga "Cefotaxime", ahakoa e kore e taea te whakaritea "Tsefasin" "Tsetaks" ranei ki te whakamahi i runga i te tikanga i runga ake. Ko te meka ko e ahu maha iwi ki arowhānui anake "kape whanaunga 'tauira matüora o te tauira taketake o whanonga, a reira te kāri rongoā tangohia e tango ki pūkete te hōtaka, me te inenga" rua "me tātai i te mātanga mātanga.

e tūtohu ana te hua taketake mō te whakamahi, ki te:

  • he manawanui pāngia ki te māuiuitanga o te pūnaha romahā i roto i te puka o te kakā, whēwhē ranei Bronchitis, me ētahi atu paturopi kahore e kawea mai te hua e hiahiatia ana;
  • taimaha te manawanui e meningitis kitakita ahu whakamua;
  • whakapumautia whakamātautau te aroaro o te endocarditis;
  • i roto i te wā postoperative i taea ki te karo i pōauautanga i te puka o te whakangaromanga wāhi o te kiri membrane o whekau faufaa me / ranei;
  • noho māngai hopuhopu iho i roto i te wheua, me werohanga intramuscular ki taero-taurite kore i mana ta'etotonu ki runga ki a ratou;
  • Gram-kino ranei karamu-pai patunga wera ngoto me mate i whakapataritari tauine (ki runga, ki te sepsis);
  • i reira ko te hiahia hoki āraihia.

tohunga Independent ahu ki te whakapono e reira he iti tetahi orotahi "Cefotaxime" taea ki te whakaatu mārama faaite dynamics pai ki te mate Lyme. Ko reira hono fakamanatu mai utu e whakaahuatia te taketake, raro ki te tono auau, me te mahi ki te fekuki maitai pai (kōrero, whakatapua ki te mita o te akoranga haumanu, kua whakanohoia tūroro i runga i te Ngā Huinga).

Whakamahi, me te inenga

(E kore e rite whai hua rite te whakatakoto he dropper werohanga, kia rite ki te tahi mau tākuta me tūroro) te tūnga hei paturopi whawhai mahi-hāngai nui mate kitakita whiriwhiri "Cefotaxime" ako. Ka rite ki whakahuatia i mua, i reira e toru iahiko kaiwhakahohe tuku: i te honikoma whaowhia jet ranei, me te roto i werohia intramuscular. ture kotahi mo te faaineineraa o te inu e mahi kore e tīariari, na ko te mea nui ki te whakatau i roto i mua i te aratau o whakahaere o te tarukino.

Manufacturer, i roto i ngā, taunaki e whai ake nei i tenei hātepe:

  • mo te werohanga / th: kia rewa 1 karamu o te paura ki te i roto i te 4 ml o te wai, lidocaine novocaine ranei;
  • hoki werohanga rō-uaua: 1 go o taonga he tika ki te tareka i te wai horomata (4 ml);
  • hoki / i roto i te e whaowhia: i roto i te pounamu ki e rua karamu cefotaxime Me ki tāpiri 100 ml o NaCl (0,9%) te taua e rima ōrau kūhuka ranei.

Tukunga kaiwhakahohe wā:

  • i / m werohanga: 5-10;
  • i / i roto i te whakataki jet: 5.3 min;
  • ka tautuhinga dropper: 50-60 min.

kawea Tātaitanga o inenga taurite, me te tabula i te hanganga o te fariiraa tino pai i roto i takitahi. E te reira ki pūkete te tau o te manawanui me te taimaha o tona tinana, kia rite ki te pai kia rite ki te momo o te mate, me te wāhanga o tona whanaketanga. I tua atu, i te menemana i hanga i roto i te hītori haumanu.

Otiia, i te tohutohu otiia whakarato pārongo i runga i reiti toharite o te tono "cefotaxime" tarukino. Werohanga (rite puehu diluted, whakaahuatia i roto i te taipitopito i runga, engari, taa, te nuinga tata katoa urupare e te whakaaro e te werohanga - he āhua mamae, me te kino te tukanga, tae noa ki nga kupu tohutohu katoa o te kaiwhakanao), i roto i ngā, kua whakaritea hoki ngā āhuatanga ngāwari, pakaru i roto i te 4-12 haora, me te horopeta kotahi o 1-2 karamu. Hoki tino me te nui subcritical i roto i tauari / whakataki (i te tere o te 2 g katoa 4 haora, engari e kore e neke atu i te 12 g / ra).

Pediatricians i roto i te talena kōwhiringa arahina e taitamariki taimaha tinana manawanui, me te tapeke tauhohe tinana ( "paerewa" - i rua ki te ono werohanga jet: 50-180 mg / kg).

pānga taha

A, no te faaue i te medicament "Cefotaxime" (e kore e rite whakapati rite honikoma whaowhia werohanga whakawākanga, mai te maha haere tahi te whakataki / m i te mamae: no te tenei take, kia rite ki te "whakarewa" Kei te nuinga o te procaine lidocaine ranei) e kore e taea te waho wāhanga mahi mohiotia o te pūnaha me whekau o te manawanui.

whakaaetia:

  • pāwera "whakautu" i roto i te puka o te nui-unahi urticaria, angioedema candidiasis ranei;
  • raruraru i te taumata o te wahi gastrointestinal (ruaki, whakapairuaki, uaua - jaundice cholestatic);
  • disorders i roto i te toto (he maturuturunga iho i roto i te tatau mōtepe, anemia hemolytic me te m. p.).

nunu'a o te tuwhena rawa

hua nui i roto i te whakaritenga o ia rā, he mahi wehe ki dysbiosis me encephalopathy; hoki pea e utua irritations kiri.

Ko te mahi tuatahi, ko te ki te whakarite kia te tuku kaiwhakahohe mutu ki te tinana. E tika ana ki te ū te āhua here ki te whakamahi o ngā hua pharmacological desensitizing (ki te aroturuki i te rata) mehua atu.

E ai ki nga contraindications kaiwhakanao

E ai ki te kōrero i homai i roto i te tauākī e pā ana, "cefotaxime" (werohanga ki tamariki, te tikanga whakaritea i muri i te taenga 30 marama o tau, i mua i paitanga ki te ahau / e whaowhia) e kore kia whakamahia:

  • i roto i te hapū;
  • hypersensitivity ki kai;
  • te tuwhera me te katinga toto;
  • Ki te māngai kē wāhanga o enterocolitis i hītori.

taunekeneke tarukino

I roto i te aratohu taketake hāngai ana ki te i te meka e kore e kia whakahaerea tahi atu rongoā i raro i tetahi huru (i tetahi pūrere rata) ki te tikanga rongoā paturopi "cefotaxime".

Werohanga (i roto i te whakamahi o te honikoma i roto i ngā o te pāhekoheko pharmacological ki ngā wāhanga o ētahi atu raau taero, he kahore rerekē i te werohanga / m), i roto i ngā, ka taea e whakapataritari kino ki nga whatukuhu, ki te "hoa" whakaahuatia faaineineraa te mahi i tetahi aminoglycoside he diuretic koropiko ranei. I roto i te tahuri, interlocks kaha tautāwhi i secretion tubular withdrawal tukanga kaitauhohe homai me whakaihiihi hua o tona kukū.

Ko te huinga ki te antiplatelet hoki houhou no o te mōrea o te toto.

tūnga ako Motuhake

"Cefotaxime" (analogs tableted, kia rite ki arotake me kōrero e iti iho whai hua) i ētahi wā whakaoho teka tauira Kumbusa me "spoofs" tātaritanga mimi mo te kūhuka pono.

A, no te kia kawea wā roa-therapy kia inea te wae hanganga o te toto i roto i kore iti iho i te 1 te wā i roto i te 10 ra.

I roto i nga ra wawe o te maimoatanga e kore e tutakina i te puka nui o te korere. A, characteristically, taua tairitenga "Cefotaxime" (mō ngā tamariki i raro i te tau o 12 tau tuku ki "piki" Kei te kore tūtohutia), rite "Fagotsef" pikitia haumanu rite ko nui iti noa.

Inu waipiro i roto i therapy i runga i te pūtake o te kaiwhakahohe te tino rāhuitia.

I te mea rite e ngákaunuitia ki "Cefotaxime" tūtohu te whakamahi o tohunga motuhake?

Comments i runga i "Sefotake" me "Tsefantrale" rite he uhinga tatau o te hua pharmacological whakaahuatia i konatunatua. Whakawa i nga arotake, ratou whakaaro te mahi atu pinepine atu i te tuhituhi i roto i tohutohu whakahaunga ki te hoko i te taua taua "Tsefabola" ranei "te pupirikana-i runga i-tono." Heoi, ahu etahi tūroro ki te whakapono e te pānga haumanu o te tauira tuku ki tautuhia ruarua me te tūponotanga o te whanaketanga o tauhohe mohiotia tuwhena tiketike.

A, no te ki te wānanga i whakaarahia te pātai kei te rite hukihuki "cefotaxime" kihai i taua i ahatia, he maha kaiwhakaako tohutohu:

  • whakamātautau, a kahore he he whakautu ki ranei te hūhi whakauru motuhake (ki te he tamau te syndrome me procaine diluted paura, ka reira he take ki te whakapono e te hūhi - he putanga o te mate pāwera, kaua ki te pānga tika o te taonga);
  • titiro hoki he rerekē tika.

Tātaritanga o whakaaro whakaatu e te nuinga o "faatura" i roto i taurite whakawhiwhia "Te Lorax." Heoi, me i mua ki te whakakapinga o tetahi matū hohe ki tetahi kōrero tonu te mātanga.

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