Hauora, Mau faaineineraa
"Betacam": tohutohu mō te whakamahi, analogs me arotake
Hei whakakore i te pēhanga tiketike, me o tini o nga mate cardiac te whakamahi i te tikanga beta1 adrenoblokatornye. Ko tētahi taua rongoā ko te tarukino "Betacam". Tohutohu mō te whakamahi whakaahua ana ia kia rite ki te tarukino e whakaaturia cardioselective, antihypertensive me sympathomimetic mahi.
Ngā āhuatanga noa
whakaaro ana tēnei taputapu te pūārai beta1-adrenergic waihanga. I whakaputahia e Kaiperu tipu "Medokemi LTD" i roto i te puka papa ki te takotoranga ma ranei nui ma paninga.
Medicament "Betacam" ako i runga i te whakaahuatanga o te faaineineraa kei roto te momo e whai ake nei: kua ratou āhua porotaka ki papa biconvex, i reira te mea he tūponotanga vahe'i Unuhia. Ki te whatiia koe i tetahi papa, na, ka waiho nga tirotiro o te ma roto tata ma ranei.
I medicament "Betacam" ako i runga i te whakaahuatanga mōkihi kiritaki he hakari te ara e whai ake nei: kia kotahi mōkihi kei toru opupu. tākai ia aratau pereti pūtau kei i 10 papa.
hanganga
I roto i te rongoā e hoatu te tūranga matua ki te wāhanga o nāianei i roto i te puka o te betaxolol hydrochloride tote. Ko te inenga o ia papa ko 0,020 g
He tikanga o "Betacam" ako i runga i te hanganga o kai hohekore fakamatala'i kahore te tauwhāiti ratou te tatau. Papa i hanga konutai glycolate starchy, te huka, te waiu, stearate konupora, microcrystalline momo cellulose, aerosil, Titanium waikura, me polyethylene glycol hydroxymethylpropylcellulose tohu 400.
tikanga o te mahi
I rongoa fakapapau'i "Betacam" ā-ako beta1 cardioselective -adrenoblokatornuyu kahore tūturu mana mahi sympathomimetic. whakaatu i te papa rawakore membrane aueue tōtika.
he tika ki te mahi e whakaiti i te putanga cardiac o te uaua ngakau, me te whakaiti i whakaongaonga kaungāongo'i i roto i te oko toto i te taha mahi Antihypertensive.
e kore e taea te huaina pānga selectivity o te raau taero i runga i te hanganga o te β 1 -adrenoreceptor herekore, no te mea kia pā pota tiketike o te betaxolol β 2 receptor hanganga -adrenozavisimye e e kei roto i te oko bronchi me te toto.
Ārai i te mahi o te raau taero, tango ki pūkete nga āhuatanga pharmacodynamic e pā ana ki te hekenga i roto i auau ngakau i okiokinga me te i roto i mahi. Ko reira e tika ana ki te inhibition o ngā β-adrenoceptor i roto i te kōpuku pakohu, e pōturi ratou automaticity.
Reira te whakaiti hoki te tuku o myocardial auheke i roto i te huru kaha, me te hāngū o te tinana, meinga nei e mauāhara whakataetae o catecholamines me mutunga karere piringa o te momo adrenergic.
te whakaiti i te raau pēhanga toto systolic me diastolic i roto i nga pera i era atu, me te i roto i te mahi, te whakaiti hua orthostatic pūpū i roto i te auau o contractions ngakau. he pānga pērā o te raau taero te whakaiti i te kawenga i runga i te myocardium.
tikanga adrenoblokatornoe Beta puai mahi antihypertensive i te huarahi e whai ake nei:
- heke putanga cardiac;
- whakakorea spasm i roto i te iatuku i te taha tika ki te mahi pokapū, e tauwhāiti te pini pukuaroha ki taiepa iaia i roto i braking mahi renin.
e kore e whakahaere wā roa o te tarukino whakaiti tona pānga hypertensive. Ki te tangohia e tatou i te horopeta kotahi betaxolol 0.005 0.04 ranei g, ka whakaatu i te whakaiti pēhanga i muri anake 3 4 ranei haora.
I roto i te rongoa, tohu "Betacam" Taupānga Kaiwhakamahi e whakahaere i te inenga 0.005g take pānga antihypertensive nei kaha ko rua ngā wā raro atu i ki te papa katoa.
Ko te mahi antihypertensive mōrahi o tetahi kukū o betaxolol puta i muri i 7-14 ra.
toketaá haumanu o medicament kore e meinga pānga cardiodepressivny motuhake, kahore pānga i runga i pākia e kūhuka, te roa e kore e whakanui i te tīhiko konutai me te inu i roto i nga kopa.
Aha whakamahia te
Drug "Betacam" ako i runga i te whakaaturanga ngā te rārangi e whai ake nei:
- pēhanga toto tiketike;
- mate te AVC uaua auheke myocardial, myocardium infarction i te tukanga;
- cardiomyopathy hypertrophic.
whakaritea te rongoā te ka i reira he huringa i roto i te ngakau, e kua whakahuatia i roto i te whakaterenga o te manawataki pakohu, tachyarrhythmias ventricular me te āhua supraventricular, roa depolarization o te myocardium, arrhythmia e pā ana ki prolapse i piha mitral, production nui o hormones thyroid.
Me pēhea te ki te whakamahi i
I rongoa "Betacam" tohutohu mō te whakamahi i peita horopeta i runga i te huru o te manawanui. inu katoa toharite horopeta ia inu. e kore e Food pā te absorption o rongoā. kia horoi iho te papa ki te wai ma.
pēhanga toto nui haere tukinotia horopeta tīmatanga rā o i 0,005 ki te 0,010 g muri 7 14 ranei ra, ki te tika, ki te whakapiki ake i te nui o medicament 0,020 g
Ko wai e kore e whakamahi i
Ehara i te katoa ka taea te whakamahi o te tikanga o "Betacam" ā-ako. Contraindications e pā ana ki te tūtohutanga nui ki nga kai, me te betaxolol hydrochloride.
E kore te whakaritea te reira no te tūroro e whai ma'i uaua ngakau puka iti hoki sinoatrialnuyu me te blockage atrioventricular i roto i te tohu tuarua, me te tuatoru, bradycardia, hypotension, arahau whakaeke huangō, angina noa.
Drugs "Betacam" papa tohutohu mō te whakamahi e kore hoki te momo inu ki ru cardiogenic, mutunga angiotrofonevroze iaia tūtohu, te whakanui ake i uaua myocardial auheke, ophthalmoplegia asthenic, endarteritis obliterans, emfizemnom lesion o pūkahukahu kikokiko, ma'i taunutia pūāhua Bronchitis huka mellitus.
huringa kitea i roto i nga whatukuhu, me te pāpaka psoriatic contraindicated te mo te maimoatanga.
tauhohe kino
pānga kino te tikanga o "Betacam" tono Kaiwhakamahi ngā mokowhiti puhoi, blockage atrioventricular, iti hoki uaua cardiac, te maturuturunga iho orthostatic i te pēhanga, tohanga rawakore huri noa te taha, ringa maha matao me waewae, paresthesia. Heoi fakahohaasi pūnaha iaia me te ngakau.
spasm arahau, hikaka, urticaria, psoriasis, kanohi maroke membrane mucous kia puta tauhohe taha me okana ataata romahā, kiri.
Ka taea e te raau meinga te momoe, huru asthenic, disorders fakalotofo'í, rohirohi nui, whakama, tohu o moemoea, te mamae āmai me te ānini.
tukanga houhou i roto i te pūnaha kūnatu e pā ana ki whakapairuaki, retching, korere, whakaroa heamana cholestasis.
Ētahi atu faaiteraa o te mahi tarukino i taea e heke o te leukocyte me ngā pūtau toto mōtepe, ka whakaiti hoki mananga.
Āhuatanga o te maimoatanga
Whakaae o tetahi tarukino kia pā ana ki etahi onäianei, e whakawhirinaki i runga i te rōpū pharmacological, te hanganga, me te inenga o te raau taero e whakamahia ana.
Rongoā "Betacam" ako i runga i te whakamahi o ngā tohutohu motuhake e hoatu mo ia take o paerewa-kore, tono whakarongo.
Na i te wā tuatahi o te maimoatanga e meinga he kore o te uaua ngakau i roto i te iwi e pängia ana ki tenei ine.
Pire "Betacam" kopare nga tohu o te kāwanatanga hypoglycemic, te nuinga o nei whakaaro ko te takahi o te manawataki cardiac. kia tango i tēnei matauranga ki tūroro pūkete e kua piki te huka toto. rapu ratou aroturuki auau o ngā taumata toto kūhuka.
Ki te whakamahi koe i taero, taunaki whakarongo ki te mana o te auau ngakau "Betacam" (papa) ako ā-ringa. I roto i te take o bradycardic disorders pakohu te manawataki, ki te inenga tika whakaiti whakakore te kaihoko maimoatanga raraunga ranei.
E titau te reira te whakamahi tupato o te tarukino i roto i te tūroro ki te mātauranga pheochromocytoma.
Ko te rongoā i ngā ki tikanga kawea e inhalation rehunga te i roto i, ai te whārua o myocardial uaua mahi auheke, me te e tukupu ana te pēhanga toto. Non-depolarizing whakaatu relaxants uaua te papa mahi auroa ka whai wāhi ki "Betacam".
Ki te hiahia koe ki te kawe i roto i te pūāhua wawaotanga hāparapara whakamaheretia, whakakore faaineineraa e rua nga ra i mua ki te kaupapa e kore nga papa i pā i te rehunga whānui.
e kore Medicament maimoatanga mutu "Betacam" ā-ako taunaki kotahi, engari āta, me te whakaiti i roto i te dosing mō te 7 14 ranei ra, ki te karo i te tauhohe o te kaiao ki whakakorenga tarukino. Nga ra e toru heke te nui o te raau taero e 0,005 g
e kore papa e tangohia ki taero e he retarders Monoamine oxidase whākōkī.
mahi Hypotensive o te tarukino me te whakaiti i estrogen nonsteroidal drugs antiinflammatory e faataere te katote konutai me te wai, engari tautāwhi i hoki te ariā o pūhui prostaglandin i te whatukuhu.
whakamahi tukutahi o diltiazem, amiodarone, me verapamil pire "Betacam" arata'i ki nui haere mahi inhibitory betaxolol hydrochloride i myocardial contractility uaua auheke me tona kawe ia.
Ko te rongoā i ngā ki cardiac taero glycosidic whakatairanga momo poraka atrioventricular.
I ngā ki ētahi atu antihypertensives faarahi papa mahi hypotensive "Betacam".
heke kukarou miramira whakaora o betaxolol i to ratou whakahaere tukutahi.
Ko te huinga o "Betacam" papa agonists xanthines ranei ai vaivai tahi o ratou mahi.
Phenothiazines me betaxolol hydrochloride mā te tauhohe i ake i tona ihirangi i roto i te toto.
Medicine "Betacam" ārai taka tango kei roto lidocaine theophylline ranei.
faarahi Sulfasalazine serum kukū o betaxolol hydrochloride.
Kāore he kōrero i runga i te whakamahi o te raau taero i roto i te tūroro pediatric.
hiahiatia tūpato kei roto i te tono o papa ki te iwi i te pei i te waka motor, me te wahine e hapu ana, me te lactating.
enei taputapu
Na roto i te beta1-adrenoblokatornym Drug Whakahaere whakarōpū rongoā "Betacam" ā-ako. no ano hoki Analogs ki tenei piha o pharmacotherapeutic. Kei roto ratou i te mahi whakauru hohe rite betaxolol hydrochloride.
whakaaro French te he tairitenga o te tarukino "Lokren", whakaputaina e "Sanofi Winthrop Ahumahi" i roto i te puka o te papa pani kiriata ma. Puka ratou a tawhio noa ki mata biconvex, i roto i nei takoto te tūpono te me te wehe i whakairo ti'araa "KE 20".
He he he horopeta kotahi o 0.02 go o betaxolol hydrochloride. wāhanga Ngaahi Houalotú rongoā ngā waiu huka, microcrystalline cellulose, konutai carboxymethyl te momo, te hauhā silicon colloidal, stearate konupora.
Ka taea te kitea te hanganga kiriata paninga hypromellose, polyethylene glycol tohu 400, Titanium hāorarua.
Drug hokona i roto i te mōkihi pepa ki e rua opupu o papa 14.
Tono rongoa ki te whakakore i te pēhanga toto tiketike, kua ngā ano reira ki atu taero ki takawhita.
Ka taea e te tarukino kawe i āraihia atu ki te whakatutuki i te exacerbation o angina i roto i te puka kukū.
te tikanga rite Russian ko te tarukino "Betaxolol", whakaputaina nei e "tipu Moscow endocrine" i roto i te puka o papa kiriata ma pani. E ratou he āhua a tawhio ki mata biconvex. whakaaro te whakauru kaha te betaxolol hydrochloride i roto i te nui o 0,020 g te wāhanga ngaahi houalotú ngā waiu huka, te konutai māngaro glycolate, aerosil dehydrated, stearate konupora, microcrystalline momo cellulose. i hanga te paninga kiriata e polyvinyl waipiro hāorarua-Titanium, talc, Macrogol 3350 waitohu, Opadry ma-2.
whakamahia ana tēnei taputapu kei te systemically ki te pēhanga toto tiketike.
He ko tetahi rongoā "" Betaxolol "i roto i te puka o pata kanohi, e kua tono topically i momo papahewa tuwhera-koki ma'i ki pēhanga intraocular tiketike, whakaora kite i muri i wawaotanga taiaho trabekuloplasticheskogo.
whakaaro o tūroro
Mō te tikanga o "Betacam" tohutohu mo te whakamahi o te mau hopearaa houhou o arotake ngā te wāhanga "tauhohe kino". e kore ai ēnei tohumate tika puta ka whakamahi i te tarukino.
Ka taea te rongo maha tūroro pai urupare e pā ana ki te beta1-adrenoblokatornom tikanga "Betacam" e maitai akono takawhita me angina. Fele tango tahi papa ki ētahi atu taero antihypertensive i roto i te therapy matatini e whakarei ake ratou whai huatanga.
maimoatanga hoki pēhanga toto Post ki noa, e nui whakapiki hauora o te manawanui.
He hoki arotake o raau taero e whakaatu te memeha noa o te maimoatanga ki tenei kaihoko.
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