HauoraMau faaineineraa

"Gabapentin" me te waipiro: arotake. "Gabapentin": tohutohu mō te whakamahi, mua manawanui me kaiwhakaako

Mai i te wā wa ki, te whakararuraru i cramps uaua maha iwi. Heoi, whakaaro ruarua iwi e pā ana ki te aha te tikanga e ara taua āhua.

E ai ki te toi, ka taea e haurangi e rerekē: te whakatakiruatanga o (toniki, clonic, toniki-clonic me myoclonic) me te kanohi (ohie, me te matatini). he tarukino whakamahia ki te hamani haurangi muri rite "Gabapentin". Ka tohutohu mō te whakamahi, arotake me contraindications o te tarukino kia te aroaro he iti i muri mai.

tonu kia tuhia te reira e, no te hukihuki wāhanga āhuatanga e te ngaro o te mate o te mahara. huru onge peheé. puta ratou haurangi āhua clonic e pā ana i te uaua ringa, waewae, me te mata.

Composition, whakaahuatanga, hua tākai me tona hanganga

hokona medicament "Gabapentin" I roto i te aha puka? pūrongo Mua e taea te hokona tenei rongoā i te rongoā i roto i te puka o capsules gelatin pakeke i roto i te ma. Ratou ihirangi Ko te tarukino ma kowhai ranei paura.

Ko te whakauru kaha o tenei kaihoko ko gabapentin. Hoki, ngā reira he taonga atu i roto i te puka o te konutai carboxymethyl māngaro, konupūmā stearate me te microcrystalline cellulose. Ka rite ki mo nga capsules, i roto ratou gelatin me Titanium hāorarua.

I roto i te mōkihi hokona te tarukino "Gabapentin"? arotake Kiritaki mea e runga i nga whata o pharmacies taea te kitea i te tarukino i roto i mōkihi pepa, e kua whakanohoia rānei capsules polymeric kēne aratau o te pūtau ranei.

Ko te parau tumu o te mahi o te tarukino

Nahea te tarukino "Gabapentin"? Tohutohu (E aroaro arotake o te rongoā i te mutunga o te tuhinga) pūrongo e te raau taero i roto i tona hanganga, ko te tino rite ki te neurotransmitter waikawa kama-aminobutyric (Kepa mo te poto). Heoi, kia tuhia te reira e te mea faufaa rerekē i te tahi atu raau taero e taunekeneke ki Kepa-receptors (hei tauira, valproate, barbiturates, benzodiazepines, o Kapa inhibitors transaminase, o Kapa inhibitors reuptake, Kepa agonists me prodrugs o o Kapa) te parau tumu o tona mahi.

He raau i Tirohia kahore āhuatanga Kepa-raa a e kore e pā te hopu me te pākia o o Kapa. Kua whakaaturia tohunga rangahau e te whakauru kaha o te kaihoko i te here ki te α2-δ-subunit o takere konupūmā ngaohiko-ti'aturi, nui te whakaiti i te rere o katote konupūmā, e tākaro he wāhi tino hira i roto i te tīmatanga o te mamae neuropathic.

Āhuatanga tarukino anticonvulsant

He aha ētahi atu āhuatanga e nohoia e te tarukino "Gabapentin"? Reviews o taote mea e he reira rawa whai hua mō te mamae neuropathic. whakaiti ana tēnei raau mate neuronal glutamate-ti'aturi, te whakanui ake i Kepa te kōtuitanga, me te te tukanga o te pehanga o te tuku, me te monoamine rōpū neurotransmitter.

E kore e taea e tatou te mea e i nohanga hauora hāngai o te tarukino "Gabapentin" e kore e herea ki receptors o ētahi atu taero (ranei neurotransmitters), tae atu ki ngā receptors Kipea, me te GABAB, me glutamate, receptors benzodiazepine, glycine, ko N-mewaro-r- aspartate.

Hāunga i "Carbamazepine" me "phenytoin", whakaaro kore e te medicament taunekeneke ki takere konutai. Te faaineineraa "gabapentin" wāhanga attenuates te pānga o te glutamate receptor agonist pērā i N-mewaro-D-aspartate. Ano, i te reira tino whakaiti te tuku o neurotransmitters monoamine.

Ko te āhuatanga konikoni o te tarukino

He aha e te tūturu neke tawhā capsules "Gabapentin"? e kore e Mua e taea ki te whakautu i tēnei pātai. Hei kitea reira, ka whai koe ki te tahuri ki ngaio mātanga tohutohu kopakia ana ranei.

E ai ki te muri, ka mea te bioavailability o kahore e hautanga ki te inenga whāngai taero. A, no te iti te nui o te tarukino te.

Ki runga ki te fariiraa i te medicament ki tona kukū wē mōrahi kitea i muri i te 3 h. Ko te bioavailability pūmau o te tarukino i roto i capsules he tata ki te 60%. Food, tae atu ki te ngako rawa, e kore pānga i runga i nga kinetics o te tarukino.

kawea Unu "Gabapentin" o toto o te manawanui i roto i te taha o te tauira rārangi. Ko motuhake o te horopeta wā hawhe-te ora, me te he āhua 5-7 haora.

Ko te āhuatanga konikoni o te tarukino kore e huri noa, ka te tono reira toutou. Ka taea te tohu i te kukū o te tarukino i roto i te toto i runga i te hua o tona whängainga kotahi.

Ko te medicament "Gabapentin" nui e kore e herea ki pūmua wē (iti iho i te 3%). Kei te whakaaturia te reira i roto i te puka tonu i nga whatukuhu.

Metabolize te rongoā e kore e kitea. Ano, e kore e reira kaha ai whākōkī oxidative ate, e whai wāhi i roto i te pākia o te tahi atu raau taero.

Ko te whakawātea o te kaihoko i te toto heke i roto i te iwi pakeke me tūroro ki te mahi tākihi waimaero.

nekehia atu faaineineraa "gabapentin" te i te tinana i te tātari toto.

Tuhinga ki te farii i rongoā

I roto i te mea mate e whakaaro tatou he tarukino ngā whai hua? He aha te iwi e mea e pā ana ki tenei urupare?

"Gabapentin" pānui pai iho i roto i:

  • mamae neuropathic i roto i tūroro pakeke (18 tau, me te pakeke);
  • monotherapy ranei rite te tarukino tautoko mo te maimoatanga o haurangi wāhanga, haere tahi i te whakatau tuarua i roto i ngā pakeke me taiohi i 12 tau o te tau.

Contraindications ki te fariiraa i rongoā

He aha e kua te tarukino contraindications "Gabapentin"? pūrongo arotake o te tono e te mea he pānga kino ki runga ki te tinana, ki te kua te rongoā kua manakohia i:

  • hypersensitivity ki tetahi o te taonga;
  • haurangi wāhanga i raro i te tau o 12 tau.

tiaki Special Ko te tikanga i whakaritea mo te hēnga o ōna whatukuhu.

Me pēhea e tango ahau i te rongoā "Gabapentin"?

Reviews (roro āwhina tenei rongoa rawa pai) kāwanatanga kia kia whakahaerea te raau anake e te tākuta mātanga, i muri i te tātaritanga tika.

tangohia waha capsules gelatin i horomia katoa, i roto i to ratou ahua. kia pau te raau ahakoa o te paraoa, horoi ki nui wai ki raro. Ki te hiahia koe ki te whakaiti i te inenga o te rongoā ki te whakakore whakakapi ranei tona orotahi, ka tenei kia meatia māmālie mo te wiki.

Maimoatanga o te mamae neuropathic i roto i ngā pakeke

Ka rite ki i roto i tenei mahi kāwanatanga rongoā whakaaro? He aha te iwi e mea e pā ana ki arotake hauora? "Gabapentin" faaite rawa tōtika ano hoki te mamae neuropathic. I roto i te penei taua huru tuatahi horopeta ia kia 900 mg. Kei te wehea nui mea ki toru nga wahi. Ki te hiahiatia, te āta nui haere te horopeta ki te mōrahi (i.e., ki runga ki te 3600 mg ia ra).

hukihuki wāhanga

Me pēhea e tango ahau i te rongoā "gabapentin" i roto i tenei mate? Kua korerotia Reviews e taea te whakaritea te taputapu e kore anake ki ngā pakeke, engari taiohi i 12 tau.

Ko te horopeta whai hua mō ngā hukihuki wāhanga whakaaro 900-2400 mg ia ra. Maimoatanga o tenei mate e taea timata ki te 300 mg o te tarukino toru nga wa te ra. I muri kia nui haere horopeta ia ki 900 mg, me te ake me te ki runga ki te 2400 mg ia ra (wehea ki toru werohanga rite).

Ko te wā wā i waenganui i pota o te tarukino i tona fariiraa, takitoru e kore e waiho ki runga ake i te 12 haora (ki te karo i te hë o hukihuki).

pānga taha

He aha tauhohe kino kia puta i roto i te tūroro te whiwhi anticonvulsant? He aha te iwi e mea e pā ana ki tenei arotake kiritaki? "Gabapentin" i roto i te maimoatanga o te mamae neuropathic taea meinga:

  • asthenia, whara kōpeka, te mamae o te localization rerekē, te mamae hoki, mate, rewharewha syndrome, ānini, taonga taimaha, edema piringa;
  • ngangau kiwi e, ataxia, mate wareware, hypoesthesia, whakama, whanoke, whakaaro waimaero, te momoe, faaati;
  • kōroke, flatulence, korere, ruaki, mangai maroke, dyspepsia, whakapairuaki, mamae puku;
  • ponana kiri;
  • hāhā o te manawa, nui korokoro;
  • mōhiti.

I roto i te maimoatanga o haurangi wāhanga, whai wāhi te tarukino ki te ahua:

  • mamae hoki, rohirohi, kirika, ānini, mate viral, edema piringa, taimaha taonga, rohirohi, ahuatanga, edema kanohi;
  • kōroke, mate niho, korere, tokopā, nui haere te hiahia, mangai maroke korokoro ranei, whakapairuaki ruaki ranei, mamae puku, bloating, anorexia, Gingivitis;
  • tohumate o te vasodilation takawhita ranei;
  • leukopenia, te purapura;
  • piere, myalgia me arthralgia;
  • mate wareware, ataxia, whakama, incoordination, korekore, dysarthria, lability aronganui, ohoroa, pau te, nystagmus, te momoe, whakaaro rerekē, faaati, uaua aitua,, whanoke, hyperkinesia; taonga, vaivai ngaro o reflexes, manukanuka, paresthesia, riri ranei;
  • abrasions, hakihaki, minamina kiri, ponana kiri;
  • mare, pharyngitis, Rhinitis, kakā;
  • mōhiti, diplopia, atarua;
  • mate mimi, paruparu.

take o te tuwhena rawa

He aha e nga tohu o te tuwhena rawa e taea ai te mea medicament? He aha e pā ana ki tenei mea te arotake? "Gabapentin" tuwhena rawa ai rua kite, whanoke, te momoe, kupu waimaero, lethargy me te korere.

Hei whakakore i taua āhua therapy symptomatic, me te te puku pārurenga horoia, ka hoatu ki a ia waro whakahohe.

Tūroro ki nui iti hoki tākihi, whakaaturia tātari toto te.

Drug "Gabapentin" me te waipiro

pūrongo tohunga Reviews e te tōtika o te raau taero whakaaro he nui rawa. Ko te mea anake i roto i te kaupapa e te tino whakarerea te manawanui te wā o tona tono te whakamahi o te ava.

Ki te ngā i te tarukino te ki waipiro, tino kia te manawanui kē tauhohe kino i te pūnaha pokapū io (hiamoe, ataxia, me ētahi atu).

taunekeneke tarukino

neke atu i te pai Drug "gabapentin" i roto i te Neuroscience, arotake o e he, e taea te kore ngā ki ngā rongoā katoa.

E ai ki nga tohutohu, whakaiti waikawa te bioavailability o te tarukino.

whakanui i taero Myelotoxicity capsules haematotoxicity "Gabapentin".

A, no te ngā ki rehunanu kore te ona pharmacokinetics ke. Heoi, ka kia kia āta aroturuki i te huinga taua tauhohenga kino pea o te pūnaha io.

medicament i Tirohia e tangohia ai te wā kotahi ki te taero antiepileptic (hei tauira, "pentobarbital", "Carbamazepine", "Phenytoin" me te waikawa valproic) me te whakawhānau-waha. I roto i tenei take, e kore ai e huri i te kinetics.

tūtohutanga motuhake

Ahakoa te meka e te syndrome withdrawal kihai i ki te takanga o hukihuki i te maimoatanga o "gabapentin" tohua e te mutunga ohorere o te maimoatanga me taero antiepileptic i roto i te iwi ki te hukihuki wāhanga taea tonu whakapataritari haehae kaha.

e kore te mea he tikanga whai hua ki te aro ki te ngaro haurangi rongoā tirohia.

Iwi e hiahia therapy matatini ki rehunanu, kia hiahia te nui haere horopeta o "gabapentin". I roto i tenei take, whakarite aroturuki tamau o te manawanui mo te whanaketanga o te momoe. I ona rongoa tautuhi horopeta kia āta iti.

A, no te ngā "gabapentin" ki ētahi atu taero anticonvulsant kua korerotia hua pai teka i roto i te faaotiraa o te pūmua i roto i te mimi te whakamahi i takai whakamātautau Ames N-Multistix SG. I roto i tenei whakaaro, mo te taua ako tūtohu te whakamahi o te tikanga rerenga motuhake i te waikawa sulfosalicylic.

ngaio Reviews me kiritaki

He pai te nuinga arotake o rata me tūroro e pā ana ki te "Gabapentin" faaineineraa. Ēnei pūrongo whakaaro e te raau tōtika akakoromaki i te mahi. Heoi, ka te ngā reira ki te waipiro maha whakawhanake nui tauhohe kino i roto i te pūnaha io.

E kore e taea e kore ki te mōhio i te meka e te withdrawal ohorere o te tarukino e taea meinga mahara tūroro kua poutoa, lethargy me te huru kino.

Kua tuhia he tokomaha te iwi e te tikanga te rōpū o tenei whai ratou he whārua me whakaaro suicidal. Ano, maha ai rongoā te whanaketanga o te pancreatitis whakapeka.

tūtohu tohunga ki maimoatanga tarukino "Gabapentin" anake i raro i te mātakitaki o te tākuta nei e taea ki te whakarite hohoro te talena haumanu rite hiahiatia.

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