Hauora, Mau faaineineraa
Ko te tarukino "Akineton": tohutohu mō te whakamahi, whakaahuatanga, arotake
Ko te taonga kaha "Akinetona" he hydrochloride biperiden. Tablet wāhi 2 mg o taonga kaha. I tua atu, ko te aroaro o wāhanga atu (te witi māngaro, māngaro potato, monohydrate reihuka, stearate konupora, microcrystalline cellulose, copovidone, konupūmā hauwai Phosphate dihydrate, talc, te wai parakore) riro te tarukino "Akineton".
Tohutohu mō te whakamahi, kōrero te whakaahua e te puka papa o te raau taero e ngā tae ma, Valium puka. I tetahi taha o te papa i reira ko te mōrea o te āhua ripeka kuiti.
1 ml o te otinga kei lactate biperiden i roto i te nui o 5 milligrams. wāhanga atu e: injecting wai, me te konutai lactate.
pānga pharmacological
biperiden whakauru Main - holinoblokator mahi pokapū.
Te pānga tā depressing te kaha ki te mahi neuronal cholinergic i roto i te striatum, i te mea te wae hanganga o te pūnaha extrapyramidal.
Te raau ai pānga ganglioblokiruyuschimi, pakeke pānga m-anticholinergic antispasmodic me āhua i te taha (antispasmodic).
tauturu Whakamahi o te tarukino faaore e alangá faaati, e whakatika i roto i te whakamahi o te raau taero cholinergic (hei tauira, pilocarpine) me catalepsy me te uaua rigidity i roto i te tūroro te whiwhi neuroleptics. He te kaha ki te kaha ai rōpū.
Pharmacokinetics
"Akineton" herea ki pūmua wē i 91-94%. Wē whakawātea ka kia 11.6 ± 0.8 ml / min / taimaha tinana kg. He horopeta kotahi o te waihanga-waha he bioavailability o e pā ana ki 33 ± 5%.
Haere ki te waiu uma.
Biperiden tino metabolized i roto i te tinana tangata. I roto i te mimi, e kore e whakaritea te taonga i roto i te puka taui. He bicycloheptane me piperidine nga metabolites nui, e he putanga i nga feces me mimi.
kawea Elliminatsiya i roto i rua ngā wāhanga, me te hawhe te ora (T 1/2) o 90 meneti i roto i te wāhanga tuatahi me te 24 haora - tuarua te wāhanga. I roto i te tūroro kaumātua, te hawhe-ora e taea ake i nui.
Tuhinga
"Akineton" whakamahia i roto i disorders extrapyramidal piri e whakahaere o etahi rongoā (neuroleptics, antipsychotics).
Ano, tohua te tarukino te mo te tātaritanga o te mate syndrome o Parkinson, parkinsonism (kaihoko e whakahaeretia ana i roto i te huinga therapy ki te turanga)
contraindications
E kore te te whakaaro o tenei tarukino whakaaturia ina e hypersensitive ki te whakauru mātātoa o te tarukino "Akineton" koe.
Tohutohu mō te whakamahi ngā e kia kia karohia te tarukino i roto i te tātaritanga o te mate i roto i te manawanui pērā i repeure whakarahi, koki-katinga papahewa, huringa taunutia i roto i te whēkau (stenosis pylorus, pararutiki Genesis ileus).
Arrhythmia, haurangi, kai uma, kaumātua, hapūtanga ko nga āhuatanga i roto i nei "Akineton" whakahaere ki te tūpato nui.
pānga taha
E whakakitea CNS pānga taha asthenia, rohirohi, lethargy, ngoikore, te kōpā, whanoke, mana'o o āwangawanga, manukanuka, waimaero mahara, whakama, moemoea, catalepsy, tarukino ti'aturiraa tarukino "Akineton".
Tohutohu mō te whakamahi korero e pā ana ki te taha-pānga me ki te wahi o te kite - mydriasis, ngangau o noho.
āhuatanga pūnaha manawa-iaia e whakaora o te auau ngakau (tachycardia); ētahi wā - whakapōturinga (bradycardia); ka tono te puka i werohia o te faaineineraa - heke i roto i te pēhanga toto (hypotension).
I runga i te wahi o te pūnaha kūnatu - mangai maroke, tohu dyspeptic, kōroke.
I runga i te wahi o te pākia e - whakaiti sweating.
I runga i te wahi o te pūnaha mimi - i roto i te tūroro ki te whakarahi (hypertrophy) o te repe repeure - uaua taea te tiana.
mate pāwera: porahurahu i runga i te kiri, minamina.
Methods o Whakamahi
Hoki intramuscular, rō-uaua, me te puka papa waha he faaineineraa pai "Akineton".
Tohutohu mō te whakamahi fokotuu e therapy "Akinetonom" te tikanga tīmata i pota iti, te horopeta atu piki stepwise rānei i runga i te pānga haumanu hiahiatia me mo ngā pānga taha.
Ngā pakeke i te whakamahi o te puka-waha o te faaineineraa tīmata maimoatanga i te horopeta o te 1 mg 1-2 fariiraa i roto i te ra 2 mg ranei wehea ki e rua pota ia ra. I tua atu, e taea te nui haere te inenga ki te 8 mg rua ki te wha pota wehea. Heoi, e kore e nui horopeta neke atu i te 2 mg ia ra. Kaua e nui ake i te inenga mōrahi tikanga 6 ki Th-16 mg mō ra rima. e kore e horopeta Single puka tarukino injectable nui 2.5-5 mg. kia korerotia tenei horopeta i muri i te hawhe haora, engari te maha o minitatanga ia ra e kore e nui ake 4 wā. Ko te horopeta mōrahi o medicament i roto i te puka injectable he 20 mg hoki nga ra e rima. A, no te tae i te horopeta tino pai te, na he whakawhitinga ki te fariiraa "Akinetona ia faataere."
Otiia e kore e wareware e pā ana ki te huarahi takitahi ki ia manawanui i roto i te therapy whakarite biperidenom.
māuiuitanga Extrapyramidal puta tika ki ingestion o etahi rongoā (antipsychotics neuroleptics ranei) titau ohipa o te taonga i homai i roto i te horopeta kotahi o 2 mg waha parenterally ranei. whakahaere tukurua o pota mea ai kia hawhe katoa haora. Heoi, ka rite ki tohua i runga ake, te maha o nga minitatanga kia kore nui ake 4 wa. kia wehewehea te horopeta-waha ki tetahi ki te e toru werohanga.
mate o Parkinson Ko tā whakahaere i te tarukino waha i 6-8 mg i roto i 2-4 pota wehea mo te ra, e taea te āta nui haere te horopeta ake ki 6-16 mg.
Tamariki i raro i te tau whakaaro kōrero te taea o te raau taero i roto i te puka injectable āta, he horopeta kotahi o te 1 mg 0.2 ml ranei. A, no te tau i te tau kotahi ki te ono tau e whakahaeretia ana 2 mg 0.4 ml ranei. Mai i 6 ki te 10 tau - 3 mg 0.6 ml ranei. kia korerotia tenei horopeta i muri i te hawhe haora ki te whawhati tata. I roto i te aroaro o ngā pānga kōaro i runga i te whakahaere o te tarukino kia werohia faahope.
I roto i te puka-waha o te therapy tarukino i roto i te tau i te 3 ki te 15 tau o tango te inenga o 1-2 mg i roto i 1-3 haora i roto i te ra.
E kore e taea e te papa inu i runga i te puku kau, a me inu e koe i te nui āhua o te wai. I takanga o ngā pānga taha houhou i te pūnaha kūnatu me tango te tarukino tonu i muri i te kai, te whakaiti i te pakeke o te pānga kino te tikanga o "Akineton".
Tohutohu mō te whakamahi tohu e i roto i te take o te nikotīni paihana i roto i ngā pakeke e whakahaerea ano therapy paerewa matatini tenei tarukino, me tona horopeta ko 5-Th-TB-10 mg mō ngā puka injectable, engari anake i roto i ngā take e whakawehi ora o te manawanui.
A, no te pau ranunga ūkuikui organic kawea dosing biperiden te i roto i takitahi i runga i te pakeke o pāpaka rānei. Tīmata i te horopeta o 5 mg i te take o te whakahaere rō-uaua, tonu whakahaere toutou noa ngaro nga tohu paihana.
tuwhena rawa
Tuwhena rawa faaite pānga anticholinergic korerotia meinga e te rongoā "Akineton".
Tohutohu mō te whakamahi, tākuta tūturu whakarongo ki te meka e te maimoatanga o tenei huru posimptomnaya (tiaki o te Cardiovascular me ngā pūnaha romahā, te hāora therapy, tūāhuruiti ako, he huinga pū tōngāmimi mimi, ki te tika). E hiahiatia ana te whakataki o te inhibitor cholinesterase (physostigmine matua) .
pāhekoheko
"Akineton" i te whakamahi o te m-holinoblokatorami, taero he he antihistamine me mahi antiepileptic whakarei faaiteraa o te muri. Heoi, tono tukutahi o metoclopramide whakaiti tona pānga haumanu. He incompatibility tarukino ení ki te waihā. piki quinidine Wāhui i roto i nga wa te mōrea o te whakawhanake i tohu dyskinesia. whakarei pānga M-cholinergic te ka tono levodopa.
Rokiroki me te hoko
Ki te hoko i tēnei tarukino titau te whakahaunga ki te whakarato i te rongoā. Hei rokiroki "Akinetona" Me ki te ū ki te pāmahana, t. Kore e E. Hauhā pāmahana nui 25 nekehanga (degrees tauine). E hinaaro tatou i te taea o ngā tamariki ki te whare "Akineton".
Manual homai te ora papa o te tarukino - rima nga tau.
Ara
Wāhui o biperiden i roto i te hapū me te whāngai ū (hohipera) titau tohu tino.
Ka taea e Biperiden tiki ki te tamaiti i roto i te waiu uma, meinga he kore rangitahi o whāngai ū ki te korenga atu o te tarukino "Akineton".
tohu whakaahuatanga Hua i roto i taua i roto i whakatau i runga i te whakarite o te biperiden i roto i te hapū, me te hohipera tango ki pūkete te tūpono ki te tamaiti, kukune.
riro kaumātua he take mōrearea mo te maimoatanga ki tenei tarukino. Na whakaritea "Akineton" tenei rōpū o te iwi ki te tūpato nui.
Kickaha ngaro o tetahi taunakitanga o te whakamahi o te haumaru i roto i te tamarikitanga, ko te take e kore e e te tono ki te tarukino tamariki "Akineton".
Whakaahuatanga o te faaineineraa (ā-ako) āta te meka e hiahiatia tūpato te ka whakamahi i tenei tarukino i roto i te tūroro ki te haurangi fibrillation ranei.
Ki te whakamahi auroa kia whakawhanake fakafalala tarukino.
Ko te mōrea o te withdrawal syndrome tā te mutunga āta o te therapy "Akinetonom".
kia te whakamahi o inu waipiro-kei roto kia karohia i roto i te therapy.
Maimoatanga ki tenei tarukino titau te nohopuku i peia waka me hākinakina ngā mahi e rapua e kukū tiketike, me ngā hohenga whakamātau tinana tere, mai e waha ana i te reira ki taua mea i te ati pea e tika ana ki te mōrea o te whanoke.
"Akineton". Tohutohu mō te whakamahi. analogs
Taurite o te faaineineraa e te matū e whai ake nei: "Biperiden" "Mendileks" "hydrochloride biperiden".
"Akineton". Reviews
Ko tino whai hua i roto i poroa te maimoatanga o tremors parkinsonism i te e alangá mo e i muri i te wā wā poto te tarukino. Ta pai-nohotahi tarukino "Akineton".
Urupare i runga i nga Ngā Huinga korero e pā ana ki te taea o te whakakitenga o te tahi mau pānga taha ia tango i te raau taero.
Utu "Akinetona". te wahi ki te hoko
Ko te utu o te otinga kia tawhio 800 moni.
Utu waihanga-waha "Akinetona" - 560-580 moni.
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