"Pyrazinamide" Papa i bactericidal pānga bacteriostatic o anti rānei i runga i te kukū ranei. tonu mahi raau te anake i raro i ngā āhuatanga waikawa (i te pH o te 5.6, me te i raro). i runga i oneone te taea rongoā whanaketanga o te ātete, i heke te tūponotanga o te whakamahi i te rongoā ki ētahi atu āpiha antitubercular. Te faaineineraa "Pyrazinamide" (fakapapau'i ako ā-tenei) he whai hua te nuinga ka te mate kohi kino rite kitea mo te wa tuatahi, tukanga momo tuberkulomah caseous-pneumonic, lymphadenitis caseous. Whakahekea te tarukino utu transportation urate me te waikawa uric, Ka taea e Hyperglycemia meinga. Ko te raau i te wahi gastrointestinal tata rawa, me te hohoro whenumi. pūmua wē herea medicament 10-20%. I muri i te haora e rua ranei, i reira ko te kukū mōrahi o moni. Kei te wehea pai rongoā i runga i te fluids tinana me te kopa, ka takoto i roto i nga whekau, tae atu i te pūkahukahu, ate, whatukuhu, me ngā wāhanga o ā pāpaka tuberculous. Founga haere te BBB. puta pākia i roto i te ate.
iteraa papû
Medicament "pyrazinamide" (whakautu o tohunga whakau reira) ko te whiriwhiri tuatahi i roto i te maimoatanga o te mate kohi.
talena dosing
I kitea te reira e kore te mea whai hua nui monotherapy. I roto i te hononga ki tenei ā-tarukino "pyrazinamide" ako taunaki ana te whakamahi i roto i ngā ki ētahi atu rongoa ki TB hohe. Hoki ngā pakeke, te inenga he 30-35 mg / kg kotahi te ra. Hoki tūroro kotahi iti iho i te rima tekau kirokaramu, te inenga ko e toru papa (1.5 g). A, no te te papatipu, ko te kia tango neke atu i te 50 kg 4 papa. (2 g). Hoki ngā tamariki i te horopeta mōrahi - 2 karamu. tangohia te raau i te kai. e tūtohu ana ki te inu i te rongoā i roto i te parakuihi.
tikanga "Pyrazinamide". Tohutohu mō te whakamahi. Ara
Medication tuwhena rawa i roto i te hanganga ture ki te whakahau a te tākuta meinga e kore. A, no te riro koe i te nui o te tarukino kitea pānga kino o te pūnaha io pokapū - whanoke, pāhoahoa me etahi atu. tuhipoka whakararuraru i roto i te ate, pea dyspepsia. Ki te whakaaturia paihana maimoatanga symptomatic. I mua a i roto i te maimoatanga TB i roto i te tūroro i runga i 60 tau kawea i roto i te aroturuki marama o tohu o bilirubin, AST, waikawa uric me te ALT. I roto i disorders o te ate titau tango o te tarukino. I roto i te tūroro ki te mate huka pea atu ki te whakawhanake e suka. A, no te ngā ki rongoā tango rongoā "Rifampicin" taea te kite hepatotoxicity. A, no te ngātahi ki te faaineineraa tono "Probenecid" pea whakaiti excretion me rite ki te hua, nui haere te tāoke. He kia kia ripeka-tūtohutanga ki rongoā "Inh", "Ethionamide" waikawa nicotinic me ētahi atu tikanga he hanganga matū rite. "Pyrazinamide" rongoā (tohutohu mō te whakamahi fakapapau'i tenei) hāngai mō rima tau. Kei te rongoa te hanganga i roto i te tākai hiri, i roto i ngā wāhi e tiakina i te marama.