Hauora, Mau faaineineraa
"Moxonidine": tohutohu mō te whakamahi, tūturu
He aha te mea te rongoa "Moxonidine"? Tohutohu mō te whakamahi o tenei taputapu, arotake e pā ana ki reira, contraindications, a kua whakaahuatia analogs i roto i te taipitopito i roto i tenei tuhinga. I tua atu, ka korero ki matou a koutou e pā ana ki te tikanga he aha e whakaaro tatou te tikanga te, ki te he ia tetahi pānga taha me te puka i roto i nei whakaputaina ai.
Ko te āhua me te hanganga o te tarukino
taea ki te hoko i te tarukino "Moxonidine" I roto i te aha puka? Ana tēnei raau e anake hokona i roto i te puka o papa. Ratou huānga kaha ko te taonga pērā i moxonidine. Ki te whakaaro ki wāhanga atu e pā ana ki taua cellulose microcrystalline, te hinu Katoro, Aerosil A-380, hydroxypropylcellulose, stearate konupora me te Tween-80.
Papa e hokona i roto i te mōkihi pepa. kia kotahi mōkihi 98, 60, 56, 42, 40, 30, 28, 20, 14 me te 10 papa.
Ko te āhuatanga pharmacological o te tarukino
He aha te mahi e hiahia ana ahau rongoā "Moxonidine"? kī Tohutohu mō te whakamahi i tenei teuteu ko te tarukino antihypertensive. Ko tōna tikanga o te mahi takoto i roto i te meka e te tikanga taonga kaha pānga te hononga pokapū i roto i te pēhanga toto ture. I roto i te mau parau te tahi atu, moxonidine - he imidazoline receptor agonist (te nuinga).
Ko te raau inhibits te mahi o te pokapū vasomotor, whakaiti i te pānga pukuaroha heke i runga i te pūnaha Cardiovascular. Ko te pēhanga (diastolic me systolic) heke āta.
He rerekē i ētahi atu āpiha sympatholytic antihypertensive medicament whakaaro e tatou i roto i taua kua reira anake te marena iti ki te Arepa-2-adrenoretseptoramm. E whakamārama ana tēnei i te tūponotanga iti o te mangai maroke me te whakarokiroki.
E kore e taea e tatou te mea e taea te whakanui ake moxonidine taiāki tūtohutanga taupū (āhua 21 ōrau) i roto i te iwi ki te mōmona.
Pharmacokinetics o te tarukino
Hea horomia te tarukino te, "Moxonidine"? tono Kaiwhakamahi kī e muri i te fariiraa i medicament tonu a tata tino whenumi i roto i te wahi kūnatu runga.
Bioavailability (pūmau) o te taputapu, ko te 88 ōrau. tutuki ana te kukū mōrahi te i muri i meneti e ono tekau ma rima. I roto i tenei take, te kohi o te kai he kahore pānga i runga i nga pharmacokinetics o te huānga hohe kua kore.
Communication ki te pūmua toto ko e pā ana ki 7.3%. Ko te metabolite nui o Moxonidine Moxonidine mahi pārōnaki dehydrated, me guanidine.
ko 150 me 300 meneti aua te hawhe-ora o moxonidine me ona metabolites.
I muri i ingestion mō te rua tekau-wha haora o te raau excreted e te whatukuhu i roto i te rōrahi o 90%. Ano, te taonga kaha mai i roto i, me te roto i te whēkau.
Tuhinga mō te whakamahi o te pūrere hauora
I roto i ētahi wā, kaitūtohu 'Moxonidine "? Ko te whakamahi o tenei raau whakaaturia anake, ki te taua māuiuitanga rite takawhita matua.
Contraindications ki te whakamahi o te pūrere hauora
I roto i ētahi wā, e kore e kaiwhakaako whakahau rongoā ki o ratou tūroro 'Moxonidine "? Tohutohu mō te whakamahi o tenei tarukino kore kei roto i te rārangi rawa roa o contraindications. Whakaaroa reira i teie nei.
Na contraindications ki te whakamahi o "Moxonidine" faaineineraa e te whai ake āhuatanga:
- faaite AV-poraka 2 me 3 nekehanga, SSS;
- bradycardia (iti iho i te 50 kapakapa ki te meneti);
- hongofulu me tau o ngā tamariki (18 tau);
- kore ngakau ma'i, me te whakapeka;
- kai pēpi wā;
- Hypersensitivity ki te huānga hohe.
Ko te tarukino "Moxonidine": tohutohu mō te whakamahi
Ka Mua e pā ana ki tenei medicament kia aroaro i te mutunga o te tuhinga. Na e hiahia ana ahau ki te korero ki a koutou e pā ana ki te pehea, ki te whakamahi i te raau tika i mua ia tatou.
Drug "Moxonidine" e roto anake. Inenga i roto i te therapy tarukino wawe kia 200 micrograms kotahi ia ra. Neke atu i te wa, ka taea e te tango e koe 400 micrograms.
E titau te reira i te whakatikatika takitahi o te nui rā o te rongoā i runga i te tolerability o therapy tarukino rānei. E ai ki nga tohutohu, te inenga mōrahi o medicament ia ra ko te 600 mg (wehea ki e rua kaupae).
Hoki tūroro ki iti hoki tākihi (āhua, me te kino), me te iwi e te hunga i runga i tātari toto, faaterehia te raau i roto i te nui o 200 mg kotahi te ra. Ki te tika (ki te manawanui pai), ka taea te nui haere te inenga i tohua ki te mōrahi (i.e. 400 mg).
pānga kino i muri i te fariiraa i medicament
E nga pānga taha o te tarukino "Moxonidine"? Mua e pā ana ki a ia e mea e te tahi mau taime te rongoā mau ai te ino o te hauora.
- pūnaha Nervous (pokapū): pāhoahoa, kaihapai, whanoke, me somnolence.
- wahi kūnatu: ruaki, mangai maroke, korere, dyspepsia me te whakapairuaki.
- pūnaha Cardiovascular: bradycardia, te maturuturunga iho tohua i roto i te pēhanga toto, hypotension orthostatic.
- Kiri, me te kiko subcutaneous disorders: edema angioneurotic, pruritus me te hikaka te kiri.
- disorders hinengaro: pau te me te ohoroa.
- Labyrinth disorders o te okana māna: waea i roto i te taringa (tupu rawa uaua).
- Musculoskeletal Pūnaha: te mamae hoki, mamae i roto i te kaki.
- pānga taha Common: edema piringa, me te asthenia.
Ka rite ki a koutou e taea te kite, e taea "Moxonidine" pire meinga ino o huru o te manawanui. Ki te korerotia nga pānga taha, kia mutu na te horopeta o rongoā.
te tikanga o te pāhekoheko ki ētahi atu taero
Ki raau taero "Moxonidine", "Moxonidine Sandoz" me ētahi atu analogues i tauturu tarukino manawanui me kihai i meinga ia kino atu, kia ratou kia tangohia anake i runga i whakahaunga. I muri i te fariiraa tukutahi o te taputapu ki ētahi atu rongoa taea meinga tauhohe e hiahiatia. He aha rite, ka titiro tatou i teie nei.
whakamahi kotahi-wā o te tarukino "moxonidine" ki te āpiha antihypertensive taua taea meinga he pānga tāpiri.
Pōuritanga (tricyclics) whakaiti i te tōtika o te raau taero antihypertensive mahi pokapū. I roto i tenei whakaaro, e kore e tūtohutia ratou mo te whakamahi i roto i te taha ki te taonga pērā i moxonidine.
whakapā i Tirohia te medicament taea ngāwari exacerbate te pānga o te raau taero, pōuritanga tricyclic, me te waihā ewaro, hypnotics me sedatives.
Ko te taonga kaha ko te medicament tika attenuated whakapiki i mahi hinengaro iwi e riro wā kotahi lorazepam.
Ahakoa kia te whakarite o "Moxonidine" raau taero, me "benzodiazepine" tūkino pärönaki whakarokiroki o te muri.
mea Tohunga e whiwhi Moxonidine e secretion tubular. I roto i te hononga ki tenei e kore kia whakamahia reira ki taero e e hoki whakanuia e secretion tubular.
Ko te wā o te hapūtanga me te hohipera (hapū me te hohipera)
Ka taea e ki te wā o te hapūtanga tango rongoā "Moxonidine-LF"? Kei Tohutohu tarukino te mōhiohio e te tino whakahaere a i whakahaeretia rawaka rangahau e pā ana ki te haumaru o rongoā whakaaro i roto i te hapūtanga. Ko te aha e kore te reira tūtohu ki te whakamahi i tenei kāwai o tūroro.
E kore e taea e tatou te mea e kore e kia whakamahia te tarukino "Moxonidine" i roto i te whāngai ū. Ko e tika ana ki te meka e te miramira te reira ki te waiu o tona whaea tenei. Ki te i roto i te hohipera tarukino ano i whakaritea, ka kia kia mutu uma-kai.
I roto i te tukanga o te rangahau (whakamātautau) i roto i nga kararehe, i kitea ai e pānga te medicament embryotoxic.
arata'iraa Motuhake i runga i te whakamahi o te rongoā
E ai ki nga tohutohu piri, i kia kia tino tupato te whakamahi o te tarukino "Moxonidine". Rawa mo reira he kāwai motuhake o tūroro. E, whakaahua tatou i teie nei.
Ngā tūpato ka tono "Moxonidine" medicament ki kia kitea i roto i te tūroro ki te AV-pā 1 tohu. Ko e tika ana ki te meka i taua iwi i reira ko he mōrea nui o bradycardia tenei.
Ano te fariiraa i te tarukino kia whakahaeretia i raro i te mātakitaki o te rata ki te nui mate te AVC, hēnga o ōna whatukuhu, me te angina iu. Tenei meka Ko e tika ana ki te meka i kore he rawaka te wheako o te whakamahi i te tarukino ki taua abnormalities.
Ki te hiahia koe ki te whakakore i te te whakamahi tukutahi o taero "moxonidine" me beta-blockers, me tuatahi whakakore koe i te parepare whakamutunga, he torutoru nga ra i muri mai - i te tuarua.
Ki te rā i reira he kore taunakitanga e arata'i tu "Moxonidine" tarukino ki te pēhanga toto nui haere. Heoi, ahakoa e otiia tūtohu tohunga ki te wāhanga i roto i te rongoā. kia te inenga kia heke i runga i te wiki e rua kua pahure.
ahakoa pānga te tarukino te kaha ki te pei nekeneke waka?
I roto i te wā o te maimoatanga hauora ki te hiahia "Moxonidine" iwi ki te kia rawa tupato ka kau i roto i ngā mahi kino, me te i te pei nekeneke waka. Ko e tika ana ki te meka e kia pokanoa te tarukino ki fariiraa tenei kukū , me te whakamātau tinana tauhohe.
Analogs, me te utu o te tarukino
Hokona te tarukino "Moxonidine" i roto i te rongoā e taea e koe, kahore whakahaunga. Ko ngā iti te utu o tenei tarukino. Per mōkihi, e kei 14 papa e whai koe ki te utu e pā ana ki 115-135 moni Russian.
Ki te whakaaro tatou he tarukino kore koutou e haere mai, ranei koutou kahore i tika i taea ki te kitea i te reira i te rongoā, i muri i tirohia ki te mātanga, takoto te muri kei te ki te tūtohu i te orotahi tarukino. I roto i enei rongoa e hiahia ana ahau ki te whakanui i te whai ake: "Fiziotenz", "Moxonidine-C3", "Moksarel", "Tumau o Moxonidine", "Moksoniteks", "Moksogamma", "Tenzotran" me pera i runga i.
kia mau ki te moni tino rite ki te kupu o te tākuta. Hoki, i mua i kia kia waia ki nga tohutohu piri te whakamahi o te rongoā.
Ko te tarukino "Moxonidine": arotake o ngā tākuta, me ngā tūroro
E ai ki ngā mātanga, he tino whai hua mō te takawhita tenei tarukino. ngā tenei whakaaro e tūroro. Heoi, amuamu etahi o ratou e muri i tango i te papa i muri i te ia faaite mai ratou pānga taha pērā i pāhoahoa, mangai maroke, pau te me te whakapairuaki. I roto i tenei take, tūtohu tākuta rongoā ki te whakakore me te whakakapi i tona orotahi, i te mea haumaru hoki hauora.
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